BDBM31883 9-cis-retinoic acid (9cRA)::ALL-TRANS-RETINOIC ACID::AT-RA::Atralin::CHEMBL38::MLS000028588::SMR000058245::TRETINOIN::Vitamin A acid::[3H]RA::[3H]Retinoic acid::[3H]Vitamin A acid::[3H]tretinoin::all-trans retinoic acid::cid_444795
SMILES C\C(\C=C\C1=C(C)CCCC1(C)C)=C/C=C/C(/C)=C/C(O)=O
InChI Key InChIKey=SHGAZHPCJJPHSC-YCNIQYBTSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 52 hits for monomerid = 31883
Affinity DataKi: 0.400nMAssay Description:Binding affinity towards cRARbeta2 receptor by displacing 1.1 nM 3[H]-9-cis-RAMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity towards cRARbeta2 receptor by displacing 0.82 nM 3[H]-all-trans-RAMore data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:Agonistic activity of the compound towards retinoic acid receptor-betaMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Binding affinity to retinoic acid receptor beta using [3H]-CD 367 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Inhibition of [3H]-ATRA binding to Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
Affinity DataKd: 13nMAssay Description:Transactivation potency of the compound was determined for Retinoic acid receptor betaMore data for this Ligand-Target Pair
Affinity DataKd: 17nMAssay Description:Inhibition of [3H]-ATRA binding to human Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
Affinity DataKd: 12nMAssay Description:Binding constant for baculovirus-expressed Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
Affinity DataEC50: 1nMAssay Description:Transcriptional activation in CV-1 cells expressing Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
Affinity DataEC50: 87nMAssay Description:Transcriptional activation in CV-1 cells expressing Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
Affinity DataEC50: 105nMAssay Description:Transcriptional activation in CV-1 cells expressing Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Binding affinity against retinoic Acid beta receptor using [3H]- -9-cis-Retinoic Acid in competitive binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.5nMAssay Description:Transcriptional activation of Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid A receptor RAR betaMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of murine Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
Affinity DataEC50: 12nMAssay Description:Effective concentration against Retinoic acid receptor betaMore data for this Ligand-Target Pair
Affinity DataEC50: 80nMAssay Description:Binding affinity against retinoic Acid beta receptors cotransfected into CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataKd: 13nMAssay Description:Binding affinity for baculovirus-expressed Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
Affinity DataKd: 0.400nMAssay Description:Apparent binding constant for Retinoic acid receptor beta in HeLa cellGAL-4 transactivation assayMore data for this Ligand-Target Pair
Affinity DataKd: 13nMAssay Description:Inhibition of [3H]-ATRA binding to baculovirus expressed Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
Affinity DataEC50: 80nMAssay Description:Transcriptional activation of Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
Affinity DataKd: 13nMAssay Description:Dissociation constant for binding to Retinoic acid receptor betaMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of binding to retinoid A receptor RAR betaMore data for this Ligand-Target Pair
Affinity DataKd: 11nMAssay Description:Effective concentration for retinoic acid recptor RAR beta transcriptional activationMore data for this Ligand-Target Pair
Affinity DataKd: 13nMAssay Description:Ability to displace 3[H]-(all-E)-retinoic acid (5 nM) from beta retinoic acid receptor (beta RAR) using transactivation assayMore data for this Ligand-Target Pair
Affinity DataKd: 13nMAssay Description:Inhibition of [3H]-RA binding to retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
Affinity DataEC50: 1.5nMAssay Description:Transcriptional activation of Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
Affinity DataKd: 7nMAssay Description:In vitro binding affinity for Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Inhibition of [3H]-ATRA-Hl60 binding to Retinoic acid receptor betaMore data for this Ligand-Target Pair
Affinity DataIC50: 0.940nMAssay Description:Binding affinity for Retinoic acid receptor betaMore data for this Ligand-Target Pair
Affinity DataKd: 11nMAssay Description:Binding affinity towards retinoic acid receptor beta was determined using [3H]-ATRA (5 nM) as radioligandMore data for this Ligand-Target Pair
Affinity DataEC50: 38nMAssay Description:Effective concentration for retinoic acid recptor RAR beta transcriptional activationMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Displacement of [11,12-3H]ARTA from RARbetaMore data for this Ligand-Target Pair
Affinity DataEC50: 12nMAssay Description:Activity at human RARbeta ligand binding domain expressed in COS7 cells cotransfected with Gal4-DBD assessed as transcriptional activation after 16 h...More data for this Ligand-Target Pair
Affinity DataEC50: 80nMAssay Description:Agonist activity for retinoic acid receptor RAR beta in transcriptional activation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.5nMAssay Description:Transcriptional activation of retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
Affinity DataEC50: 1.5nMAssay Description:Transcriptional activation for RAR beta receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 80nMAssay Description:Transactivation potency of the compound was determined for Retinoic acid receptor betaMore data for this Ligand-Target Pair
Affinity DataEC50: 1nMAssay Description:Compound was tested for functional activity in CV-1 cells transfected with an expression vector for retinoic acid receptor beta using transactivation...More data for this Ligand-Target Pair
Affinity DataEC50: 6.31nMAssay Description:Agonist activity at RARbeta2 expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
Affinity DataEC50: 25.1nMAssay Description:Activity at RARbeta1 expressed in mouse NIH3T3 cells by R-SAT assayMore data for this Ligand-Target Pair
Affinity DataKd: 13nMAssay Description:Compound was tested for functional activity in CV-1 cells transfected with an expression vector for retinoid X receptor beta using transactivation as...More data for this Ligand-Target Pair
Affinity DataEC50: 78nMAssay Description:Transcriptional activation in CV-1 cells expresing human Retinoid X receptor RXR-alphaMore data for this Ligand-Target Pair
Affinity DataEC50: 38nMAssay Description:Ability to inhibit TTNPB-induced transactivation at retinoic acid receptor alphaMore data for this Ligand-Target Pair
Affinity DataEC50: 0.520nMAssay Description:Transactivation of mouse Gal4-fused RARbeta-LBD expressed in COS-7 cells after 1 day by bright-Glo reagent based assayMore data for this Ligand-Target Pair
Affinity DataEC50: 18nMAssay Description:Transactivation of GST-tagged RARbeta LBD (unknown origin) assessed as fluorescein-labelled coactivator peptide recruitment measured after 4 hrs by T...More data for this Ligand-Target Pair
Affinity DataEC50: 25nMAssay Description:Transcriptional activity against RARbeta1More data for this Ligand-Target Pair
Affinity DataEC50: 6.30nMAssay Description:Transcriptional activity against RARbeta2More data for this Ligand-Target Pair
Affinity DataKd: 13nMAssay Description:Inhibition of [3H]-ATRA binding to baculovirus expressed RAR beta receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 38nMAssay Description:Agonist activity RARbeta (unknown origin) assessed as induction of receptor transactivationMore data for this Ligand-Target Pair